From: Antibody-drug conjugates: integrated bioanalytical and biodisposition assessments in lead optimization and selection
Dose
(mg/kg)
t1/2
(day)
Cmax
(μg/mL)
CL
(mL/day/kg)
Vss
(mL/kg)
AUC0-INF
(day*μg/mL)
10
3.75
90.0
195
589
51.4
3
3.42
27.8
70.3
295
42.7
1
3.90
12.0
39.8
197
25.2
0.3
3.97
2.72
31.5
170
9.52